RSC Advances
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ARTICLE
DOI: 10.1039/C5RA06935A
Biochemistry 1997, 36, 15670; (
Perlman, and M. C. Gershengorn, Bioorg. Med. Chem.
2002, 10, 189; ( ) N. Kaur, X. Lu, M. C. Gershengorn, and
R. Jain, J. Med. Chem. 2005, 48, 6162; ( ) N. Kaur, V.
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b) R. Jain, J. Singh, J. H.
GPCR
Gꢀprotein coupled receptor
BLAST Basic Local Alignment Search Tool
Erap1 Endoplasmic reticulum aminopeptidase 1
c
d
Acknowledgements
e
* Corresponding author. Tel. +91 (172) 2292024; Fax: +91 (172)
2214692; Email: rahuljain@niper.ac.in
6
f
Dr. Chhuttan L. Meena acknowledges the support provided by Dr.
Marvin C. Gershengorn NIDDK, NIH, USA for this study. This study
was supported by Rajiv Gandhi National Fellowship Award (RGNF)
2006, University grant commission (UGC), New Delhi, India and
Fulbright Nehru Doctrol and Professoinal Research Fellowship (FNꢀ
DPR), United State India Education Foundation (USIEF,
1493/DPR/2011ꢀ2012).
aDepartment of Medicinal Chemistry, National Institute of
Pharmaceutical Education and Research, Sector 67, S.A.S. Nagar, 160
062, Punjab, India
,
g
h
Nandekar, B. Wahlang, N. Shaikh, Y. B. Pawar, C. L. Meena, A.
T. Sangamwar, R. Jain, K. B. Tikoo, and A. K. Bansal, Mol.
Pharmaceutics 2012, 9, 2458; (i) P. Bagul, K. S. Khomane, S. S.
Kesharwani, P. Pragyan, P. P. Nandekar, C. L. Meena, A. K.
Bansal, R. Jain, K. B. Tikoo, and A. T. Sangamwar, J. Mol.
Recognit. 2014, 27, 609.
bDepartment of Pharmacology and Toxicology, National Institute of
Pharmaceutical Education and Research, Sector 67, S.A.S. Nagar, 160
062, Punjab, India
15.
16.
17.
K. S. Khomane, C. L. Meena, R. Jain and A. K. Bansal,
Expert Opin. Ther. Pat., 2011, 21, 1673.
J. A. Kelly, G. R. Slator, K. F. Tipton, C. H. Williams and
K. Bauer, J. Biol. Chem., 2000, 275, 16746.
G. A. Scalabrino, N. Hogan, G. R Slator, D. J. Gregg, C.
M. Fitchett, S. M. Draper, G. W Bennett, P.M. Hinkle, K.
Bauer, C. H. Williams, K. F. Tipton, and J. A. Kelly,
cDepartment of
Pharmacoinformatics, National Institute
of
Pharmaceutical Education and Research, Sector 67, S.A.S. Nagar, 160
062, Punjab, India
Electronic Supplementary Information (ESI) available: Complete spectral
1
data, H, 13C, HPLC of all peptides and tables depicting effect of 6c on
Neuropharmacology, 2007,
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(a
functional observation battery (FOB). See DOI: 10.1039/b000000x/
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