- Lactam glycogen phosphorylase inhibitors and method of use
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A compound of formula I wherein W is a bicyclic hetroaryl of the structure X is —O—, —S—, —SO2—, —CHR5—, —CHR5O—, —CHR5S—, —CHR5SO2—, —CHR5CO— or —CH2CHR5—;
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Page/Page column 39
(2010/02/05)
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- A versatile synthesis of 2-substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepine-3-ones
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A mild and general strategy for the synthesis of 2-substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepine-3-ones is described. The seven-membered lactam is prepared by intramolecular amide bond formation from the intermediate amino acid, which is obtained e
- Van Rompaey, Karolien,Van Den Eynde, Isabelle,De Kimpe, Norbert,Tourwé, Dirk
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p. 4421 - 4432
(2007/10/03)
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