61293-32-1Relevant articles and documents
Design and synthesis of potent N1-substituted indole melatonin receptor agonists.
Tsotinis, Andrew,Eleutheriades, Andreas,Hough, Katherine,Sugden, David
, p. 382 - 383 (2003)
The design and expeditious synthesis of two new indole analogs with up to 5-fold potency of that of melatonin is described.
Convenient modification of the Leimgruber-Batcho indole synthesis: Reduction of 2-nitro-p-pyrrolidinostyrenes by the FeCl3-activated carbon-N2H4H2O system
Taydakov,Dutova,Sidorenko,Krasnoselsky
experimental part, p. 425 - 434 (2012/01/13)
A new catalytic system containing ferric chloride, activated carbon, and hydrazine has been proposed for the reductive cyclization of β-dialkylamino-2-nitrostyrenes to give the corresponding indoles (Leimgruber-Batcho synthesis). Various substituted indoles may be obtained in high yield under these conditions.
