1373214-94-8Relevant articles and documents
Synthesis and evaluation of aryl-naloxamide opiate analgesics targeting truncated exon 11-associated μ opioid receptor (MOR-1) splice variants
Majumdar, Susruta,Subrath, Joan,Le Rouzic, Valerie,Polikar, Lisa,Burgman, Maxim,Nagakura, Kuni,Ocampo, Julie,Haselton, Nathan,Pasternak, Anna R.,Grinnell, Steven,Pan, Ying-Xian,Pasternak, Gavril W.
, p. 6352 - 6362 (2012/09/22)
3-Iodobenzoylnaltrexamide 1 (IBNtxA) is a potent analgesic acting through a novel receptor target that lack many side-effects of traditional opiates composed, in part, of exon 11-associated truncated six transmembrane domain MOR-1 (6TM/E11) splice variant