1001068-45-6Relevant articles and documents
Methodology for the preparation of 2-argininylbenzothiazole
Kenney, Birdella D.,Breslav, Michael,Chang, Rosie,Glaser, Roland,Harris, Bruce D.,Maryanoff, Cynthia A.,Mills, John,Roessler, Armin,Segmuller, Brigitte,Villani Jr., Frank J.
, p. 9798 - 9801 (2007)
(Chemical Equation Presented) An efficient process to produce kilogram quantities of a key argininylbenzo[d]thiazole intermediate was developed for the preparation of the tryptase inhibitor RWJ-56423. A variety of activated arginine esters and benzo[d]thi