diethyl 2-(aziridin-1-yl)butanedioate

Base Information

• Chemical Name: diethyl 2-(aziridin-1-yl)butanedioate
• CAS No.: 1137-24-2
• Molecular Formula: C₁₀H₁₇NO₄
• Molecular Weight: 215.249
• Mol file: 1137-24-2.mol

Synonyms:1-Aziridinesuccinicacid, diethyl ester (6CI,7CI,8CI); Butanedioic acid, 1-aziridinyl-, diethylester (9CI); NSC 24023

Chemical Property of diethyl 2-(aziridin-1-yl)butanedioate

Chemical Property:

• Vapor Pressure: 0.00267mmHg at 25°C
• Boiling Point: 286.2°Cat760mmHg
• Flash Point: 126.9°C
• Density: 1.157g/cm³

Purity/Quality:

99.5% ^*data from raw suppliers

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

SDS file from LookChem

Useful:

Technology Process of diethyl 2-(aziridin-1-yl)butanedioate

There total 2 articles about diethyl 2-(aziridin-1-yl)butanedioate which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

ethyleneimine (151-56-4,9002-98-6) + Diethyl maleate (141-05-9) → 1-<1,2-bis(carbethoxy)ethyl>aziridine (1137-24-2)

Guidance literature:

With sodium methylate;

Reference yield:

ethyleneimine (151-56-4,9002-98-6) + diethyl Fumarate (623-91-6) → 1-<1,2-bis(carbethoxy)ethyl>aziridine (1137-24-2)

Guidance literature:

With sodium methylate;

Reference yield: 80.0%

1-<1,2-bis(carbethoxy)ethyl>aziridine (1137-24-2) + Thiosalicylic acid (147-93-3) → o--2-aminoethylthio>benzoic Acid (94509-73-6)

Guidance literature:

In methanol; for 2h; Ambient temperature;

DOI:10.1007/BF00503597

upstream raw materials:

ethyleneimine

Diethyl maleate

diethyl Fumarate

Downstream raw materials:

o--2-aminoethylthio>benzoic Acid