Tetrahedron p. 304 - 311 (2016)
Update date:2022-08-02
Topics:
Kashiwa, Mitsuhiro
Kuwata, Yoshiyuki
Sonoda, Motohiro
Tanimori, Shinji
An Oxone-mediated transition-metal-free oxidative C-N bond formation has been achieved for the regioselective synthesis of substituted pyrazoles. The reactions accompany the chelation-controlled ortho-oxidation of N-substituted aromatic ring to provide ph
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